| Compounds |
ID50 with 0.5% FBS |
ID50 with 2% FBS |
LD50 |
| ID50<<LD50 |
|
|
|
| Roscovitine |
1.23 |
7.50 |
- |
| Y-27632 |
4.40 |
6.06 |
- |
| Tyrphostin AG879 |
5.91 |
8.19 |
- |
| Ethacrynic acid |
2.64 |
10.0 |
- |
| Metrifudil |
6.09 |
10.0 |
- |
| N6-(2-Amino-phenyl)ethyladenosine |
9.65 |
10.0 |
- |
| N6-Cyclohexyladenosine |
10.0 |
10.0 |
- |
| Nitrendipine |
9.65 |
10.0 |
- |
| Wortmannin |
10.0 |
10.0 |
- |
| ID50<LD50 |
|
|
|
| H-7 |
5.78 |
9.65 |
>10.0 |
| Sodium pravastatin |
10.0 |
10.0 |
>10.0 |
| Simvastatin |
2.07 |
4.04 |
>10.0 |
| BQ-123 |
3.56 |
8.93 |
>10.0 |
| BQ-788 |
3.05 |
7.88 |
>10.0 |
| LY294002 |
3.98 |
10.0 |
>10.0 |
| CGS15943 |
2.28 |
3.00 |
>10.0 |
| 15-Deoxy prostaglandin J2 |
3.21 |
7.33 |
>10.0 |
| ID50>LD50 |
|
|
|
| CP55940 |
2.51 |
6.80 |
7.84 |
| BIM I |
2.57 |
3.40 |
7.21 |
| Chelerythrine chloride |
0.49 |
0.44 |
0.52 |
| Ouabain |
0.06 |
0.36 |
0.07 |
| Okadaic acid |
0.08 |
0.07 |
0.05 |
| |
|
|
(x10-6 M) |
- : not determined |