Product Drug Indication Current status
ABI-007 (Abraxane®) Albumin-paclitaxel nanoparticle Oncology Marketed
99mTc-Albures 99mTc –aggregated albumin Oncology Marketed
99mTc-Nanocoll 99mTc –aggregated albumin Oncology Marketed
Vasovist® Albumin-binding Gadolinium (III) complex Oncology Marketed
B-22956/1 Albumin-binding Gadolinium (III) complex Oncology Marketed
Levenir® Albumin-binding fatty acid derivative of insulin Diabetes Marketed
Liraglutide (Victoza®) Albumin-binding fatty acid derivative of GLP-1 Diabetes Marketed
Albuferon® Albumin-fusion protein of interferon-α-2b Hepatitis C Phase III
AT-103 (Ozoralizumab) Albumin-binding nanobody directed against human TNF-α Rheumatology Phase II
INNO-206 Albumin binding prodrug of doxorubicin Oncology Phase II
ABI-008 Albumin-docetaxel nanoparticle Oncology Phase II
MTX-HSA Methotrexate albumin conjugate Oncology Phase I/II
MM-111 Albumin fusion protein directed against ErbB2 and ErbB3 Oncology Phase I/II
AFL-HSA Albumin conjugate of aminofluorescein Oncology Phase I/II
CjC-1134-PC Albumin conjugate of exendin-4 Diabetes Phase I/II
ABI-009 Albumin-rapamycin nanoparticle Oncology Phase I
ABI-010 Albumin nanoparticle with a HSP90 inhibitor Oncology Phase I
Table 1: Albumin-based drugs or imaging agents on market and under clinical trials.