Substrates Inhibitors Inducers
Antipsychotics:
Asenapine
Clozapine
Haloperidol
Olanzapine
Chlorpromazine
Fluphenazine
Pimozide
   
Antidepressants:
Amitriptyline
Clomipramine
Duloxetine
Fluvoxamine
Imipramine
Mirtazapine
Fluoxetine
Fluvoxamine
Paroxetine
Sertraline
 
Others:
Caffeine
Diazepam
Melatonin
Phenacetin
Tacrine
Theophylline
R-warfarin
Zolpidem
  Amiodarone
Caffeine *
Ciprofloxacin
Enoxacin
Ginkgo biloba  
Cigarrette smoke
Barbiturates
Carbamazepine
Phenytoin
Rifampicin
Ritonavir
Griseofulvin
Omeprazole
Lansoprazole
Table 3: Main substrates and clinically relevant inhibitors or inducers of human CYP1A2.