Substrates Inhibitors Inducers
Antipsychotics:
Aripiprazole
Clozapine
Olanzapine
Risperidone
Thioridazine
Pimozide
Quetiapine
Zuclophentixol
Asenapine
Chlorpromazine
Fluphenazine
Levomepromazine
Perphenazin
Haloperidol
 
Antidepressants:
Mirtazapine
Desvenlafaxine
Bupropion
Duloxetine
Fluoxetine
Paroxetine
Sertraline
Citalopram
Escitalopram
Fluvoxamine
Tricyclics
Venlafaxine
 
Others:
Antiarrhythmics
Beta blockers
Opioids
Tramadol
Atomoxetine
Donepezil
Galantamine
Phenformin
Melatonin
Methadone
Amiodarone
Lansoprazole
Quinidine
Cocaine
Ritonavir
Valproicacid
Carbamazepine
Dexamethasone
Phenytoin
Rifampicin
Table 4: Main substrates and clinically relevant inhibitors, and inducers of human CYP2D6.