Transporter |
Location |
Transporter kinetics |
Reference |
PMAT |
Intestine |
Km= 1.32 mM |
[13] |
OCT1 |
Liver |
Km=1.47mM
Vmax =396pmol/min/mg protein |
[17] |
OCT2 |
Kidney |
Km=0.99mM,
Vmax =1444pmol/min/mg protein |
[17] |
MATE1 |
Liver and Kidney |
Km= 0.78mM,
Vmax = 4.46nmol/min/mg protein |
[16] |
MATE-K2 |
Kidney |
Km= 1.98mM,
Vmax = 1.69nmol/min/mg protein |
[16] |
|