IC50 (nM)  
Compound hSGLT1 hSGLT2 GLUT1 UGEa (mg/day)
Canagliflozin 910 2.2 >10000 3696
Table 4: hSGLT1, hSGLT2, Facilitated Glucose Transporter 1 (GLUT1) Inhibitory
Activity, and Rat Urinary Glucose Excretion (UGE) Data for Canagliflozin [41].