Fullerene Derivative

A23187 + FD* 48/80 + FD* somatostatin +FD* poly-L-lysine + FD*
Biotin no Inh no Inh 44.6 (±1.8)¥¥¥ no Inh
C70-OH 19.0 (±1.1)¥¥¥ 42.0 (±4.6)¥¥¥ 13.4 (±5.2)¥ 33.4 (±5.5)¥¥¥
CCC no Inh no Inh 23.8 (±0.8)¥¥¥ no Inh
DMAE 18.6  (±7.9)¥ 16.9 (±10.)¥¥¥ 24.3 (±9.7)¥ no Inh
Ethanolamine 36.0 (±3.0)¥¥¥ no Inh no Inh no Inh
Niacin no Inh 59.5 (±1.3)¥¥¥ 21.9 (±13.8)¥ 20.9 (±12.6)¥
NSAID 21.1 (±11.4)¥ no Inh no Inh no Inh
PC4 no Inh no Inh 21.6 (±2.9)¥¥¥ no Inh
Tetraglutamate 22.3 (±3.9)¥¥¥ no Inh 20.3 (±4.5)¥¥ 17.9 (±13.1)¥
Tetrainositol no Inh no Inh 32.8 (±1.9)¥¥¥ no Inh
Tetraphosphate 18.9 (±0.4)¥¥¥ no Inh no Inh no Inh
Tetrapyridine 14.0 (±1.9)¥¥ 34.8 (±8.1)¥¥ no Inh 13.1 (±4.0)¥
Tetrasulfonate 21.1 (±6.3)¥ 44.8 (±11.2)¥¥ 22.0 (±5.50)¥¥ 26.7 (±2.3)¥¥
TGA  49.8 (±8.9)¥¥¥ no Inh 16.7 (±3.8)¥¥¥ 43.8 (±10.6)¥¥
TTA no Inh no Inh 34.6 (±2.6)¥¥¥ 52.4 (±4.3)¥¥¥
* FD Treatment at 10 μg/mL. ¥¥¥ p value < 0.01 / ¥¥ p value < 0.02 / ¥ p value < 0.05 / no Inh = no significant inhibition observed
Table 1: Mean % inhibition of degranulation (±SD) in FD treated and untreated MC.