| Immunosuppressive Agent |
Year Introduced |
Category |
| Predisone |
1955 |
Glucocorticoid |
| Azathioprine |
1968 |
Antiproliferative |
| Cyclosporine |
1983 |
Calcineurin Inhibitor |
| Tacrolimus |
1994 |
Calcineurin Inhibitor |
| Mycophenolatemofetil (MMF) |
1995 |
Antiproliferative |
| Basiliximab |
1998 |
IL-2 Receptor Antibody |
| Sirolimus |
1999 |
Antiproliferative |
| Belatacept |
2011 |
Costimulation blocker |
|