Drug |
Solubility |
Absorption Characteristics (BA=Bioavailability) |
Isoniazid |
8 |
Readily absorbed (BA=91%) |
Stavudine |
12 |
Apparently fast absorption (BA 86-100%) |
Lamivudine |
14 |
BA >82% |
Doxycycline Hyclate |
20 |
>95% |
Ciprofloxacin |
33 |
Rapid absorption (BA ˜ 70) |
Levofloxacin |
40 |
Rapid (BA˜100%) |
Ranitidine |
40 |
Rapidly absorbed (BA 50-60%) |
Zidovudine |
50 |
Rapidly and almost completely absorbed |
Pyrazinamide |
67 |
Fully absorbed |
Acetaminophen |
68 |
Readily absorbed (BA=62%–89%) |
Cimetidine |
88 |
Rapidly, yet incompletely (BA 56-68%) |
Metronidazole |
100 |
Rapidly absorbed with BA >90% |
Ibuprofen |
571 |
Rapid and complete (BA 100%) |
Acyclovir |
714 |
Erratic (BA 10 to 30%) |
Rifampicin |
714 |
Well absorbed (BA ˜93%) |
Atenolol |
1010 |
Incomplete absorption, (BA 40-60%) |
Acetazolamide |
1389 |
rapidly and almost completely |
Quinine |
2000 |
Rapidly and almost completely absorbed |
Prednisolone |
4348 |
Rapidly absorbed (BA >75–98%) |
Metoclopramide |
5000 |
Rapid absorption (BA 30-100%). |
Prednisone |
8333 |
Rapidly absorbed (BA 80–100%) |
Propranolol |
16207 |
Almost completely absorbed (>90%) |
Furosemide |
54795 |
Fairly rapidly absorbed (BA 60–70%) |
Choroquine |
94340 |
Rapidly and almost completely (BA ˜ 89%) |
Efavirenz |
100000 |
Absorption? (BA 40-45%?) |
Ketoprofen |
100000 |
Readily absorbed (BA=92%) |
Verapamil |
223714 |
Rapidly and almost completely (BA 10-20%) |
Diclofenac |
421941 |
Rapid and complete (BA ˜ 60%) |
Amitriptyline |
500000 |
Well absorbed (BA ˜ 48%) |
Amodiaquine |
>1000000 (?) |
Readily absorbed |