Type of ABC transporter |
Researcher, year |
Inhibitors from natural sources |
P-gp |
|
|
|
Kitagawa et al., 2005 |
Acacetin, Galangin, Myricetin, Morin, Biochanin A and Kaempferol6 |
|
Critchfieldet al., 1994 |
Apigenin, Fisetin, Rutin7 |
|
Zhu et al., 2001 |
Tea polyphenols8 |
BCRP inhibitors |
|
|
|
Imai et al., 2004 |
Phytoestrogens (Flavonoids)9 |
|
Ahmed-Belkacemet al., 2007
Shuzhonget al., 2004 |
Bioeravinones G and H (two rotenoids) from Boerhaavia rotenoids10 Apigenin, Biochanin, Chrysin, Daidzein, Epigallocatechin (EGC), epigallocatechin-3-gallate (EGCG), Fisetin, Genistein, Hesperetin, Kaempferol, Luteolin, Morin, Myricetin, Naringenin, Naringin, Phloretin, Phloridzin, Quercetin, Silibin, Silymarin5 |
|