Receptors |
Re-docking |
OH derivative |
OCH3 derivative |
Ei |
Ki |
Ei |
Ki |
Ei |
Ki |
3QS1 |
-9.3 |
0.15 |
-8.2 |
0.96 |
-8.1 |
1.14 |
1LS5 |
-8.1 |
1.14 |
-7.5 |
3.13 |
-7.0 |
7.29 |
1SME |
-8 |
1.35 |
-7.8 |
1.89 |
-7.7 |
2.24 |
|
Ei=Binding affinity (Kcal/mol);Ki=Inhibition constant (µM) |
Table 2: Docking score results for malaria receptors. |