DNMT inhibitors Status of Clinical trial
SGI-110 Preclinical evaluation in progress
RG108 Preclinical evaluation in progress
SGI-1027 Preclinical evaluation in progress
MG98 Preclinical evaluation in progress
5-fluoro-2-deoxycytidine Phase I
5-Azacytidine (Vidaza) Completed; US FDA approved
Decitabine (Dacogen) Completed; US FDA approved
Table 2: DNA demethylating agents in clinical development
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