PARAMETER

TEST

REFERENCE

MEAN

C.V.

MEAN

C.V.

Cmax (ng/mL)

1760.5

26.6

1779.4

25.8

Tmax (hours)

3.67

26.4

3.67

39.0

AUC0-T (ng·h/mL)

30946.5

28.0

31073.6

25.7

AUC 0-∞(ng·h/mL)

31912.5

28.2

32270.9

26.4

AUCT/∞ (%)

97.05

1.6

96.49

2.3

Kel (hours-1)

0.0507

18.4

0.0503

17.3

T½el (hours)

14.07

16.6

14.18

17.1

Table 1: The Pharmacokinetic Parameters of Imatinib tablets 400mg versus Glivec.
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