Vehicle Drug Solubility (mg/mL)
Water 0.00397
PEG 400 71.6 ± 1.45
1- methyl- 2-pyrrolidinone 458.4
Labrasole 61.0
Tween 80 49.7 ± 0.41
Tween 20 55.8 ± 0.87
Cremophore EL 46.0 ± 0.69
Plurooleique CC 497 1.04 ± 0.02
Labrafac CC 1.04 ± 0.01
Caproyl 90 5.42 ± 0.06
Peanut Oil 2.19
Paraffin Oil 0.009
Linseed Oil 0.79
Lavender Oil 1.23
Corn Oil 0.42
Mineral Oil 0.004
Soybean Oil 0.31
Olive Oil 0.22
Coriander Oil 0.74
Table 1: Solubility of etravirine in various medium at room temperature.
Goto home»