Compound Concentration Range Reference
Geldanamycin 50 nM in culture [75]
AT13387 10-1000 nM  in culture [76]
SNX5422 15-250 nM  in culture [77]
STA9090 1-250 nM in culture [78]
Celastrol 0.2-10 µM  in culture [79]
BIIB021 0-250 nM in culture, 40 mg/kg in vivo [80,81]
AUY922 10- 500 nM in culture, 20 mg/kg in vivo [82,83]
Table 2: Hsp90 inhibitors currently under investigation
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